ERK5-IN-1
| Chemical Name | ERK5-IN-1 |
|---|---|
| CAS Number | 1234479-76-5 |
| MDL Number | MFCD18642659 |
| Molecular Formula | C25H29N7O2 |
| Molecular Weight | 459.54 |
Introduction of 1234479-76-5 :
ERK5-IN-1 is a potent ERK5 inhibitor with an IC50 of 87±7 nM. ERK5-IN-1 also inhibits LRRK2[G2019S] with an IC50 of 26 nM. IC50 & Target: IC50: 87±7 nM (ERK5), 26 nM (LRRK2[G2019S])[1] In Vitro: ERK5-IN-1 (Compound 5) exhibits a cellular EC50 for inhibiting epidermal growth factor (EGF) induced ERK5 autophosphorylation of 0.19±0.04 μM[1].
| Purity | NLT 98% |
|---|---|
| Storage | at 20ºC 2 years |
*The above information is for reference only.