Chemical Name |
Derenofylline |
CAS Number |
251945-92-3 |
MDL Number |
MFCD12756289 |
Molecular Formula |
C18H20N4O |
Molecular Weight |
308.38 |
Synonyms |
SLV 320 |
Introduction of 251945-92-3 :
Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1]. IC50 & Target: Ki: 1 nM (adenosine A1 receptor)[1].
Purity |
NLT 98% |
Storage |
at 20ºC 2 years |
*The above information is for reference only.