Chemical Name | SB-277011 |
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CAS Number | 215803-78-4 |
MDL Number | MFCD08690601 |
Molecular Formula | C28H30N4O |
Molecular Weight | 438.56 |
Synonyms | SB-277011A |
SB-277011 is a potent and delective dopamine D3 receptor antagonist (pKi values are 8.0, 6.0, 5.0 and <5.2 for D3, D2, 5-HT1D and 5-HT1B respectively); brain penetrant. IC50 value: 8.0 (pKi) Target: D3 receptor
Purity | NLT 98% |
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Storage | at 20ºC 2 years |