PD 151746
| Chemical Name | PD 151746 |
|---|---|
| CAS Number | 179461-52-0 |
| MDL Number | MFCD03453564 |
| Molecular Formula | C11H8FNO2S |
| Molecular Weight | 237.25 |
Introduction of 179461-52-0 :
PD151746 is a calpain inhibitor, shows a 20-fold selectivity for u-calpain (Ki = 0.26 ± 0.03 μM) over m-calpain (Ki = 5.33 ± 0.77 μM). IC50 value: 0.26 ± 0.03 μM (Ki, for μ-calpain), 5.33 ± 0.77 μM (Ki, for m-calpain) [1] Target: calpain in vitro: The μ-calpain inhibitor PD 151746 decreases oxLDL-induced cytotoxicity. [2]
| Purity | NLT 98% |
|---|---|
| Storage | at 20ºC 2 years |
*The above information is for reference only.