Chemical Name | Darusentan |
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CAS Number | 171714-84-4 |
MDL Number | MFCD00949063 |
Molecular Formula | C22H22N2O6 |
Molecular Weight | 410.42 |
Synonyms | Lu-135252 |
Darusentan is a selective endothelin A (ETA) receptor antagonist. Darusentan competes for radiolabeled endothelin binding in rat aortic vascular smooth muscle cells (RAVSMs) membranes with single-site kinetics, exhibiting a Ki=13 nM[1].
Purity | NLT 98% |
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Storage | at 20ºC 2 years |