GR 103691
| Chemical Name | GR 103691 |
|---|---|
| CAS Number | 162408-66-4 |
| MDL Number | MFCD00936840 |
| Molecular Formula | C30H35N3O3 |
| Molecular Weight | 485.62 |
Introduction of 162408-66-4 :
GR 103691 is a potent, selective dopamine D3 receptor antagonist with a Ki value of 0.4 nM. GR 103691 shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites[1]. IC50 & Target: Ki: 0.4 nM (Human dopamine D3 receptor)[1] In Vitro: GR 103691 shows marked affinity for serotonin1A (5-HT1A) receptors (Ki of 5.8 nM) and α-1 adrenoceptors (Ki of 12.6 nM)[1].
| Purity | NLT 98% |
|---|---|
| Storage | at 20ºC 2 years |
*The above information is for reference only.