L-371,257
| Chemical Name | L-371,257 |
|---|---|
| CAS Number | 162042-44-6 |
| MDL Number | MFCD00944944 |
| Molecular Formula | C28H33N3O6 |
| Molecular Weight | 507.58 |
Introduction of 162042-44-6 :
L-371,257 is an orally bioavailable, non-blood-brain barrier penetrant, selective and competitive antagonist of oxytocin receptor (pA2=8.4) with high affinity at both the oxytocin receptor (Ki=19 nM) and vasopressin V1a receptor (Ki=3.7 nM)[1][2]. IC50 & Target: Ki: 19 nM (oxytocin receptor), 3.7 nM (vasopressin V1a receptor)[2]
| Purity | NLT 98% |
|---|---|
| Storage | at 20ºC 2 years |
*The above information is for reference only.