Chemical Name | DMP-543 |
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CAS Number | 160588-45-4 |
MDL Number | MFCD00934500 |
Molecular Formula | C26H18F2N2O |
Molecular Weight | 412.43 |
Synonyms | XR-543 |
DMP-543 (XR-543) is a KV7 channel blocker, also acts as a potent neurotransmitter release enhancer[1][2]. IC50 & Target: KV7 channel In Vitro: DMP-543 enhances [3H]ACh release from rat brain slices, with an EC50 of 700 nM[2].
Purity | NLT 98% |
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Storage | at 20ºC 2 years |