Tilapertin
| Chemical Name | Tilapertin |
|---|---|
| CAS Number | 1000690-85-6 |
| Molecular Formula | C20H21F3N2O2 |
| Molecular Weight | 378.39 |
| Synonyms | AMG747 |
Introduction of 1000690-85-6 :
Tilapertin is an oral inhibitor of glycine transporter type-1 (GlyT1). IC50 & Target: GlyT1[1] In Vivo: Tilapertin is a nanomolar potent, orally bioavailable and selective GlyT1 inhibitor. Oral administration of Tilapertin dose-dependently increases cerebrospinal fluid (CSF) glycine concentration in rats[1].
| Purity | NLT 98% |
|---|---|
| Storage | at 20ºC 2 years |
*The above information is for reference only.